2013

    Fisetin: A Dietary Antioxidant for Health Promotion

    Khan N, Syed DN, Ahmad N, Mukhtar H

    Published in Antioxidants & Redox Signaling

    Abstract

    Comprehensive review of fisetin covering antioxidant properties, anti-inflammatory effects, neuroprotection, and senolytic activity. Discusses mechanisms including SIRT1 activation and multiple signaling pathway modulation.

    Methodology

    Narrative review of preclinical in vitro and animal studies.

    Key Findings

    Reviews preclinical evidence that fisetin acts as an antioxidant and anti-inflammatory flavonoid, modulating SIRT1, NF-kB, PI3K/Akt and mTOR signalling, with neuroprotective and anticancer activity in cell and animal models. Typical dietary intake is far below the doses used experimentally, and oral bioavailability is poor.

    Conclusions

    Fisetin shows broad mechanistic promise in laboratory models, but no human efficacy data support supplementation.

    Limitations

    Narrative review of in vitro and animal work only; no controlled human trials, and effective concentrations in cell models often exceed achievable plasma levels.

    Supplements Studied

    Fisetin
    Compound

    Reviews preclinical evidence that fisetin acts as an antioxidant and anti-inflammatory flavonoid, modulating SIRT1, NF-kB, PI3K/Akt and mTOR signalling, with neuroprotective and anticancer activity in cell and animal models. Typical dietary intake is far below the doses used experimentally, and oral bioavailability is poor.

    Outcomes Measured

    Reviews preclinical evidence that fisetin acts as an antioxidant and anti-inflammatory flavonoid, modulating SIRT1, NF-kB, PI3K/Akt and mTOR signalling, with neuroprotective and anticancer activity in cell and animal models. Typical dietary intake is far below the doses used experimentally, and oral bioavailability is poor.

    Study Details

    Year:2013
    Quality Score:4/10

    Disclosures

    Funding

    United States National Institutes of Health grants (University of Wisconsin authors).

    This information is for educational purposes only. Always consult a healthcare professional before starting any supplement regimen.