systematic_review
    2020

    Senolytic drugs: from discovery to translation

    Kirkland JL, Tchkonia T

    Published in Journal of Internal Medicine

    Methodology

    Narrative review of senolytic drug discovery, mechanisms and early human translation, covering dasatinib, quercetin, fisetin and navitoclax

    Key Findings

    Senolytics transiently disable senescent-cell anti-apoptotic pathways and delay or alleviate multiple age-related disorders in preclinical models; human evidence remains early stage.

    Conclusions

    Senolytics are a promising but still translational class; clinical benefit in humans is not yet established.

    Limitations

    Narrative review rather than systematic; heavy reliance on animal data; author conflicts in senolytic development.

    Supplements Studied

    Quercetin
    Compound

    The first senolytic drugs Dasatinib, Quercetin, Fisetin and Navitoclax were discovered using a hypothesis-driven approach.

    Fisetin
    Compound

    The first senolytic drugs Dasatinib, Quercetin, Fisetin and Navitoclax were discovered using a hypothesis-driven approach.

    Outcomes Measured

    Senolytics transiently disable these SCAPs, causing apoptosis of those SC with a tissue-destructive SASP.

    Study Details

    Year:2020
    Quality Score:6/10

    Disclosures

    Funding

    NIH extramural

    This information is for educational purposes only. Always consult a healthcare professional before starting any supplement regimen.