2006

    The Flavonoid Fisetin Promotes ERK-Dependent Long-Term Potentiation and Enhances Memory

    Maher P, Akaishi T, Abe K

    Published in Proceedings of the National Academy of Sciences

    Abstract

    Study demonstrating fisetin enhances memory through ERK-dependent long-term potentiation. Shows neuroprotective effects and memory improvement in aging mice, suggesting potential for cognitive decline prevention.

    Methodology

    Preclinical study combining rat hippocampal slice electrophysiology with in vivo object-recognition memory testing in mice, plus cell-culture work on ERK/CREB signalling.

    Key Findings

    Fisetin activated the ERK-CREB signalling pathway in cultured neurons, facilitated long-term potentiation in rat hippocampal slices, and improved object-recognition memory in mice given oral fisetin. Effects were blocked by MEK inhibitors, confirming ERK dependence.

    Conclusions

    Fisetin enhances hippocampal long-term potentiation and memory in rodents through ERK-dependent signalling, establishing a mechanistic rationale for investigating it as a cognitive agent.

    Limitations

    Entirely preclinical; no human data. Fisetin has low oral bioavailability in humans, so rodent dosing does not translate directly. Object-recognition memory in mice is a limited proxy for human cognition.

    Supplements Studied

    Fisetin
    Compound

    Fisetin activated the ERK-CREB signalling pathway in cultured neurons, facilitated long-term potentiation in rat hippocampal slices, and improved object-recognition memory in mice given oral fisetin. Effects were blocked by MEK inhibitors, confirming ERK dependence.

    Outcomes Measured

    Fisetin enhances memory through ERK-dependent long-term potentiation and shows neuroprotective effects and memory improvement in aging mice.

    Study Details

    Year:2006
    Quality Score:3/10

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